eBook: Formulation Technologies and Strategies for Successful New Product Development - 39

Formulation 1
Table 3: Ingredients for formulations 1 and 2 used to test drug release kinetics.
Amount (mg/tablet)
Parteck® ODT excipient
Paracetamol (acetaminophen)
Trimyristin
Silicon dioxide, highly dispersed
Total
Formulation 2
Parteck® ODT excipient
Paracetamol (acetaminophen)
Sodium stearyl fumarate
Silicon dioxide, highly dispersed
Total
700.0
250.0
40.0
10.0
1050.0
Amount (mg/tablet)
222.3
257.7
15.0
5.0
500
Compression force (kN)
Tablet thickness (mm)
Tablet weight (mg)
Table 4: Physical data for paracetamol tablets based on Parteck® ODT excipient.
20
5.0
Weight variation (%RSDa
Tablet strength (N)
)
Hardness variation (%RSDa
Disintegration (s)
Friabilityb
(%)
a Relative standard deviation | b
Friability according to the Ph.Eur./USP test method
Table 4. Physical data for paracetamol tablets based on Parteck® ODT.
Stability is Essential
In addition to examining disintegration and
dissolution properties immediately after
production, the stability of ODT formulations and
their performance over their shelf-life must be
evaluated. As the composition of some excipient
systems is not disclosed it is sometimes difficult to
foresee possible instabilities in the final formulation
due to the potential presence of impurities. Since
excipient systems for ODT formulations are usually
a combination of two or more components, their
composition can be ambiguous to the formulator.
Among the commonly observed impurities in
solid dose excipients are peroxides. Therefore, the
peroxide content in the five ODT excipient systems
)
992.8
0.49
162
15.33
44-56
0.31
Amount (%/tablet)
70.0
25.0
4.0
1.0
100
Amount (%/tablet)
44.5
51.5
3.0
1.0
100
10
4.7
498.2
0.16
172
8.66
34-54
0.25
39

eBook: Formulation Technologies and Strategies for Successful New Product Development

Table of Contents for the Digital Edition of eBook: Formulation Technologies and Strategies for Successful New Product Development

eBook: Formulation Technologies and Strategies for Successful New Product Development - 1
eBook: Formulation Technologies and Strategies for Successful New Product Development - 2
eBook: Formulation Technologies and Strategies for Successful New Product Development - 3
eBook: Formulation Technologies and Strategies for Successful New Product Development - 4
eBook: Formulation Technologies and Strategies for Successful New Product Development - 5
eBook: Formulation Technologies and Strategies for Successful New Product Development - 6
eBook: Formulation Technologies and Strategies for Successful New Product Development - 7
eBook: Formulation Technologies and Strategies for Successful New Product Development - 8
eBook: Formulation Technologies and Strategies for Successful New Product Development - 9
eBook: Formulation Technologies and Strategies for Successful New Product Development - 10
eBook: Formulation Technologies and Strategies for Successful New Product Development - 11
eBook: Formulation Technologies and Strategies for Successful New Product Development - 12
eBook: Formulation Technologies and Strategies for Successful New Product Development - 13
eBook: Formulation Technologies and Strategies for Successful New Product Development - 14
eBook: Formulation Technologies and Strategies for Successful New Product Development - 15
eBook: Formulation Technologies and Strategies for Successful New Product Development - 16
eBook: Formulation Technologies and Strategies for Successful New Product Development - 17
eBook: Formulation Technologies and Strategies for Successful New Product Development - 18
eBook: Formulation Technologies and Strategies for Successful New Product Development - 19
eBook: Formulation Technologies and Strategies for Successful New Product Development - 20
eBook: Formulation Technologies and Strategies for Successful New Product Development - 21
eBook: Formulation Technologies and Strategies for Successful New Product Development - 22
eBook: Formulation Technologies and Strategies for Successful New Product Development - 23
eBook: Formulation Technologies and Strategies for Successful New Product Development - 24
eBook: Formulation Technologies and Strategies for Successful New Product Development - 25
eBook: Formulation Technologies and Strategies for Successful New Product Development - 26
eBook: Formulation Technologies and Strategies for Successful New Product Development - 27
eBook: Formulation Technologies and Strategies for Successful New Product Development - 28
eBook: Formulation Technologies and Strategies for Successful New Product Development - 29
eBook: Formulation Technologies and Strategies for Successful New Product Development - 30
eBook: Formulation Technologies and Strategies for Successful New Product Development - 31
eBook: Formulation Technologies and Strategies for Successful New Product Development - 32
eBook: Formulation Technologies and Strategies for Successful New Product Development - 33
eBook: Formulation Technologies and Strategies for Successful New Product Development - 34
eBook: Formulation Technologies and Strategies for Successful New Product Development - 35
eBook: Formulation Technologies and Strategies for Successful New Product Development - 36
eBook: Formulation Technologies and Strategies for Successful New Product Development - 37
eBook: Formulation Technologies and Strategies for Successful New Product Development - 38
eBook: Formulation Technologies and Strategies for Successful New Product Development - 39
eBook: Formulation Technologies and Strategies for Successful New Product Development - 40
eBook: Formulation Technologies and Strategies for Successful New Product Development - 41
eBook: Formulation Technologies and Strategies for Successful New Product Development - 42
eBook: Formulation Technologies and Strategies for Successful New Product Development - 43
eBook: Formulation Technologies and Strategies for Successful New Product Development - 44
https://www.nxtbookmedia.com