eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 25

and NSP8 viral proteins. The RdRp TR-FRET Assay
kit is designed to measure RdRp-mediated
direct incorporation of biotinylated ATP into a
double-stranded RNA substrate. The increase in
TR-FRET signal is proportional to the amount of
ATP incorporated in the RNA. This assay is ideal for
high-throughput screening of enzyme inhibitors,
to perform kinetic studies, or to accurately measure
a drug EC50
.
Conclusion
TR-FRET is an ultra-low background technique
allowing the measure of any reaction in which
two labeled entities come in proximity. The main
drawback of the technique is that it requires two
optimized labeled entities, in addition to a low
dynamic range. However, these drawbacks are
offset by several advantages:
* Small volumes
* Homogeneous: no need for washing
steps or for physical separation from the
unbound entities
* Robust, sensitive signal
*
Ultra-low background with high signal to
noise ratio
Figure 6: Simple Operation
* Stable signal: use of lanthanide donor
fluorophores minimizes photobleaching
The growing commercial availability of ready-touse
TR-FRET immunoassay kits has opened the
technique to mainstream use. BPS Bioscience
offers over 80 assay kits for drug discovery in the
TR-FRET format with new products developed
regularly. Optimized, validated, high-quality assay
kits ensure reliable results, quickly.
25

eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development

Table of Contents for the Digital Edition of eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development

eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 1
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 2
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 3
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 4
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 5
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 6
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 7
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 8
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 9
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 10
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 11
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 12
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 13
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 14
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 15
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 16
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 17
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 18
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 19
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 20
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 21
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 22
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 23
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 24
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 25
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 26
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 27
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 28
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 29
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 30
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 31
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 32
eBook: Biochemical and Cell-Based Assays for Targeted Cancer Drug Discovery and Development - 33
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